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Assay Detail

CHEMBL5518342

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Binding
Inhibition of mushroom tyrosinase by spectrophotometric method
6
Total Activities
6
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Agaricus bisporus
Confidence 5 — Multiple protein complex / RNA
Curated By Autocuration

Target

Mushroom tyrosinase (CHEMBL6066154)
Type PROTEIN FAMILY
Organism Agaricus bisporus

Publication

Recent advances in triazoles as tyrosinase inhibitors.
Mermer A, Demirci S.
Eur J Med Chem (2023) 259 : 115655 -115655
PubMed 37482020 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 6 7.97 9.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL5430416 1 9.00
CHEMBL5426437 1 9.00
CHEMBL5408010 1 9.00
CHEMBL5414043 1 7.85
CHEMBL5427541 1 7.72
CHEMBL5422809 1 5.25

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL5430416 IC50 = 1.0 nM 9.00
CHEMBL5426437 IC50 = 1.0 nM 9.00
CHEMBL5408010 IC50 = 1.0 nM 9.00
CHEMBL5414043 IC50 = 14.0 nM 7.85
CHEMBL5427541 IC50 = 19.0 nM 7.72
CHEMBL5422809 IC50 = 5620.0 nM 5.25