Assay Detail
Functional
CHEMBL5521859
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Antiviral activity against DENV-1 TC974#666 infected in african green monkey Vero cells incubated for 24 hrs measured after 3 days post infection by RT-PCR analysis
24
Total Activities
22
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | dengue virus type 1 |
| Cell Type | Vero |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Discovery of JNJ-1802, a First-in-Class Pan-Serotype Dengue Virus NS4B Inhibitor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 24 | 8.52 | 10.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3905772 | — | — | 1 | 10.00 |
| CHEMBL5314530 | MOSNODENVIR | 2.0 | 1 | 9.70 |
| CHEMBL5562312 | — | — | 1 | 9.52 |
| CHEMBL5555759 | — | — | 1 | 9.40 |
| CHEMBL3923294 | — | — | 1 | 9.40 |
| CHEMBL3895322 | — | — | 2 | 9.05 |
| CHEMBL5566989 | — | — | 1 | 9.00 |
| CHEMBL3905304 | — | — | 1 | 8.70 |
| CHEMBL3889668 | — | — | 2 | 8.70 |
| CHEMBL5566158 | — | — | 1 | 8.70 |
| CHEMBL5559307 | — | — | 1 | 8.70 |
| CHEMBL5556494 | — | — | 1 | 8.52 |
| CHEMBL5559826 | — | — | 1 | 8.40 |
| CHEMBL5563912 | — | — | 1 | 8.40 |
| CHEMBL5555250 | — | — | 1 | 8.10 |
| CHEMBL5558438 | — | — | 1 | 8.10 |
| CHEMBL5555341 | — | — | 1 | 7.92 |
| CHEMBL5542636 | — | — | 1 | 7.40 |
| CHEMBL5566578 | — | — | 1 | 7.40 |
| CHEMBL4214447 | — | — | 1 | 7.07 |
| CHEMBL5563352 | — | — | 1 | 7.06 |
| CHEMBL5542213 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3905772 | — | EC50 | = | 0.1 | nM | 10.00 |
| CHEMBL5314530 | MOSNODENVIR | EC50 | = | 0.2 | nM | 9.70 |
| CHEMBL5562312 | — | EC50 | = | 0.3 | nM | 9.52 |
| CHEMBL5555759 | — | EC50 | = | 0.4 | nM | 9.40 |
| CHEMBL3923294 | — | EC50 | = | 0.4 | nM | 9.40 |
| CHEMBL3895322 | — | EC50 | = | 0.9 | nM | 9.05 |
| CHEMBL3895322 | — | EC50 | = | 0.97 | nM | 9.01 |
| CHEMBL5566989 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL5559307 | — | EC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3905304 | — | EC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3889668 | — | EC50 | = | 2.0 | nM | 8.70 |
| CHEMBL5566158 | — | EC50 | = | 2.0 | nM | 8.70 |
| CHEMBL5556494 | — | EC50 | = | 3.0 | nM | 8.52 |
| CHEMBL5559826 | — | EC50 | = | 4.0 | nM | 8.40 |
| CHEMBL5563912 | — | EC50 | = | 4.0 | nM | 8.40 |
| CHEMBL5555250 | — | EC50 | = | 8.0 | nM | 8.10 |
| CHEMBL5558438 | — | EC50 | = | 8.0 | nM | 8.10 |
| CHEMBL5555341 | — | EC50 | = | 12.0 | nM | 7.92 |
| CHEMBL3889668 | — | EC50 | = | 20.0 | nM | 7.70 |
| CHEMBL5542636 | — | EC50 | = | 40.0 | nM | 7.40 |
| CHEMBL5566578 | — | EC50 | = | 40.0 | nM | 7.40 |
| CHEMBL4214447 | — | EC50 | = | 86.0 | nM | 7.07 |
| CHEMBL5563352 | — | EC50 | = | 88.0 | nM | 7.06 |
| CHEMBL5542213 | — | EC50 | - | — | - |