Assay Detail
Functional
CHEMBL5521862
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Antiviral activity against DENV-4 H241 infected in african green monkey Vero cells incubated for 24 hrs measured after 3 days post infection by RT-PCR analysis
20
Total Activities
20
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | dengue virus type 4 |
| Cell Type | Vero |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Discovery of JNJ-1802, a First-in-Class Pan-Serotype Dengue Virus NS4B Inhibitor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 20 | 6.89 | 7.96 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5562312 | — | — | 1 | 7.96 |
| CHEMBL5314530 | MOSNODENVIR | 2.0 | 1 | 7.96 |
| CHEMBL3905772 | — | — | 1 | 7.96 |
| CHEMBL5555759 | — | — | 1 | 7.82 |
| CHEMBL3923294 | — | — | 1 | 7.36 |
| CHEMBL5559307 | — | — | 1 | 7.28 |
| CHEMBL5566989 | — | — | 1 | 7.15 |
| CHEMBL3905304 | — | — | 1 | 7.08 |
| CHEMBL5566158 | — | — | 1 | 7.02 |
| CHEMBL5559826 | — | — | 1 | 7.00 |
| CHEMBL5542636 | — | — | 1 | 6.96 |
| CHEMBL5563912 | — | — | 1 | 6.96 |
| CHEMBL5556494 | — | — | 1 | 6.96 |
| CHEMBL5558438 | — | — | 1 | 6.77 |
| CHEMBL5555341 | — | — | 1 | 6.64 |
| CHEMBL5555250 | — | — | 1 | 6.54 |
| CHEMBL5566578 | — | — | 1 | 6.12 |
| CHEMBL5563352 | — | — | 1 | 5.75 |
| CHEMBL4214447 | — | — | 1 | 5.58 |
| CHEMBL5542213 | — | — | 1 | 4.85 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5562312 | — | EC50 | = | 11.0 | nM | 7.96 |
| CHEMBL5314530 | MOSNODENVIR | EC50 | = | 11.0 | nM | 7.96 |
| CHEMBL3905772 | — | EC50 | = | 11.0 | nM | 7.96 |
| CHEMBL5555759 | — | EC50 | = | 15.0 | nM | 7.82 |
| CHEMBL3923294 | — | EC50 | = | 44.0 | nM | 7.36 |
| CHEMBL5559307 | — | EC50 | = | 53.0 | nM | 7.28 |
| CHEMBL5566989 | — | EC50 | = | 71.0 | nM | 7.15 |
| CHEMBL3905304 | — | EC50 | = | 83.0 | nM | 7.08 |
| CHEMBL5566158 | — | EC50 | = | 95.0 | nM | 7.02 |
| CHEMBL5559826 | — | EC50 | = | 100.0 | nM | 7.00 |
| CHEMBL5542636 | — | EC50 | = | 110.0 | nM | 6.96 |
| CHEMBL5563912 | — | EC50 | = | 110.0 | nM | 6.96 |
| CHEMBL5556494 | — | EC50 | = | 110.0 | nM | 6.96 |
| CHEMBL5558438 | — | EC50 | = | 170.0 | nM | 6.77 |
| CHEMBL5555341 | — | EC50 | = | 230.0 | nM | 6.64 |
| CHEMBL5555250 | — | EC50 | = | 290.0 | nM | 6.54 |
| CHEMBL5566578 | — | EC50 | = | 760.0 | nM | 6.12 |
| CHEMBL5563352 | — | EC50 | = | 1800.0 | nM | 5.75 |
| CHEMBL4214447 | — | EC50 | = | 2600.0 | nM | 5.58 |
| CHEMBL5542213 | — | EC50 | = | 14000.0 | nM | 4.85 |