Assay Detail
Binding
CHEMBL5524628
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of CPT1B (unknown origin) in KB cells
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | KB |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Carnitine O-palmitoyltransferase 1, muscle isoform (CHEMBL2216739) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Modulators for palmitoylation of proteins and small molecules.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 3 | 6.76 | 7.80 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2216778 | — | — | 1 | 7.80 |
| CHEMBL2216779 | — | — | 1 | 7.68 |
| CHEMBL2216771 | — | — | 1 | 4.80 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2216778 | — | IC50 | = | 16.0 | nM | 7.80 |
| CHEMBL2216779 | — | IC50 | = | 21.0 | nM | 7.68 |
| CHEMBL2216771 | — | IC50 | = | 16000.0 | nM | 4.80 |