Assay Detail
Functional
CHEMBL5526165
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at human AMY3R complex of CTR/RAMP3 expressed in Baby hamster kidney cells incubated for 3 hrs followed by medium replacement without compound measured after 30 mins by luciferase reporter assay
23
Total Activities
23
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Tissue | Kidney |
| Cell Type | Baby hamster kidney cell |
| Confidence | 7 — Homologous single protein target |
| Curated By | Autocuration |
Target
Amylin receptor AMY3; CALCR/RAMP3 (CHEMBL2111190) ↗| Type | PROTEIN COMPLEX |
| Organism | Homo sapiens |
Publication
NN1213 - A Potent, Long-Acting, and Selective Analog of Human Amylin.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 23 | 9.56 | 10.33 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5567107 | — | — | 1 | 10.33 |
| CHEMBL5560328 | — | — | 1 | 9.82 |
| CHEMBL5567446 | — | — | 1 | 9.79 |
| CHEMBL5567377 | — | — | 1 | 9.75 |
| CHEMBL5563010 | — | — | 1 | 9.74 |
| CHEMBL5568431 | — | — | 1 | 9.73 |
| CHEMBL5568414 | — | — | 1 | 9.70 |
| CHEMBL5568471 | — | — | 1 | 9.66 |
| CHEMBL5568545 | — | — | 1 | 9.66 |
| CHEMBL5554990 | — | — | 1 | 9.65 |
| CHEMBL5560790 | — | — | 1 | 9.57 |
| CHEMBL5566453 | — | — | 1 | 9.51 |
| CHEMBL5565993 | — | — | 1 | 9.50 |
| CHEMBL5556440 | — | — | 1 | 9.47 |
| CHEMBL5560524 | — | — | 1 | 9.46 |
| CHEMBL5566450 | — | — | 1 | 9.45 |
| CHEMBL5561117 | — | — | 1 | 9.44 |
| CHEMBL5555676 | — | — | 1 | 9.41 |
| CHEMBL5568143 | — | — | 1 | 9.37 |
| CHEMBL5532322 | — | — | 1 | 8.97 |
| CHEMBL5531967 | — | — | 1 | 8.81 |
| CHEMBL2103758 | PRAMLINTIDE | 4.0 | 1 | - |
| CHEMBL3989767 | CALCITONIN SALMON | 4.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5567107 | — | EC50 | = | 0.047 | nM | 10.33 |
| CHEMBL5560328 | — | EC50 | = | 0.151 | nM | 9.82 |
| CHEMBL5567446 | — | EC50 | = | 0.161 | nM | 9.79 |
| CHEMBL5567377 | — | EC50 | = | 0.177 | nM | 9.75 |
| CHEMBL5563010 | — | EC50 | = | 0.18 | nM | 9.74 |
| CHEMBL5568431 | — | EC50 | = | 0.186 | nM | 9.73 |
| CHEMBL5568414 | — | EC50 | = | 0.2 | nM | 9.70 |
| CHEMBL5568471 | — | EC50 | = | 0.219 | nM | 9.66 |
| CHEMBL5568545 | — | EC50 | = | 0.217 | nM | 9.66 |
| CHEMBL5554990 | — | EC50 | = | 0.222 | nM | 9.65 |
| CHEMBL5560790 | — | EC50 | = | 0.267 | nM | 9.57 |
| CHEMBL5566453 | — | EC50 | = | 0.31 | nM | 9.51 |
| CHEMBL5565993 | — | EC50 | = | 0.319 | nM | 9.50 |
| CHEMBL5556440 | — | EC50 | = | 0.34 | nM | 9.47 |
| CHEMBL5560524 | — | EC50 | = | 0.35 | nM | 9.46 |
| CHEMBL5566450 | — | EC50 | = | 0.352 | nM | 9.45 |
| CHEMBL5561117 | — | EC50 | = | 0.364 | nM | 9.44 |
| CHEMBL5555676 | — | EC50 | = | 0.39 | nM | 9.41 |
| CHEMBL5568143 | — | EC50 | = | 0.432 | nM | 9.37 |
| CHEMBL5532322 | — | EC50 | = | 1.061 | nM | 8.97 |
| CHEMBL5531967 | — | EC50 | = | 1.535 | nM | 8.81 |
| CHEMBL2103758 | PRAMLINTIDE | EC50 | = | 0.005 | nM | - |
| CHEMBL3989767 | CALCITONIN SALMON | EC50 | = | 0.0016 | nM | - |