Assay Detail
Functional
CHEMBL5526166
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity at human CTR expressed in Baby hamster kidney cells incubated for 3 hrs followed by medium replacement without compound measured after 30 mins by luciferase reporter assay
23
Total Activities
23
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Tissue | Kidney |
| Cell Type | Baby hamster kidney cell |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
NN1213 - A Potent, Long-Acting, and Selective Analog of Human Amylin.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 23 | 8.65 | 10.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2103758 | PRAMLINTIDE | 4.0 | 1 | 10.15 |
| CHEMBL5567107 | — | — | 1 | 9.50 |
| CHEMBL5560790 | — | — | 1 | 9.17 |
| CHEMBL5563010 | — | — | 1 | 9.16 |
| CHEMBL5554990 | — | — | 1 | 8.88 |
| CHEMBL5531967 | — | — | 1 | 8.86 |
| CHEMBL5568414 | — | — | 1 | 8.86 |
| CHEMBL5568431 | — | — | 1 | 8.70 |
| CHEMBL5555676 | — | — | 1 | 8.66 |
| CHEMBL5567446 | — | — | 1 | 8.61 |
| CHEMBL5568545 | — | — | 1 | 8.60 |
| CHEMBL5560328 | — | — | 1 | 8.60 |
| CHEMBL5568471 | — | — | 1 | 8.59 |
| CHEMBL5566453 | — | — | 1 | 8.58 |
| CHEMBL5565993 | — | — | 1 | 8.52 |
| CHEMBL5567377 | — | — | 1 | 8.28 |
| CHEMBL5556440 | — | — | 1 | 8.28 |
| CHEMBL5561117 | — | — | 1 | 8.26 |
| CHEMBL5560524 | — | — | 1 | 8.19 |
| CHEMBL5532322 | — | — | 1 | 8.08 |
| CHEMBL5568143 | — | — | 1 | 8.00 |
| CHEMBL5566450 | — | — | 1 | 7.74 |
| CHEMBL3989767 | CALCITONIN SALMON | 4.0 | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2103758 | PRAMLINTIDE | EC50 | = | 0.07 | nM | 10.15 |
| CHEMBL5567107 | — | EC50 | = | 0.314 | nM | 9.50 |
| CHEMBL5560790 | — | EC50 | = | 0.672 | nM | 9.17 |
| CHEMBL5563010 | — | EC50 | = | 0.697 | nM | 9.16 |
| CHEMBL5554990 | — | EC50 | = | 1.322 | nM | 8.88 |
| CHEMBL5531967 | — | EC50 | = | 1.371 | nM | 8.86 |
| CHEMBL5568414 | — | EC50 | = | 1.38 | nM | 8.86 |
| CHEMBL5568431 | — | EC50 | = | 1.993 | nM | 8.70 |
| CHEMBL5555676 | — | EC50 | = | 2.19 | nM | 8.66 |
| CHEMBL5567446 | — | EC50 | = | 2.477 | nM | 8.61 |
| CHEMBL5568545 | — | EC50 | = | 2.522 | nM | 8.60 |
| CHEMBL5560328 | — | EC50 | = | 2.492 | nM | 8.60 |
| CHEMBL5568471 | — | EC50 | = | 2.579 | nM | 8.59 |
| CHEMBL5566453 | — | EC50 | = | 2.609 | nM | 8.58 |
| CHEMBL5565993 | — | EC50 | = | 3.005 | nM | 8.52 |
| CHEMBL5567377 | — | EC50 | = | 5.21 | nM | 8.28 |
| CHEMBL5556440 | — | EC50 | = | 5.204 | nM | 8.28 |
| CHEMBL5561117 | — | EC50 | = | 5.459 | nM | 8.26 |
| CHEMBL5560524 | — | EC50 | = | 6.5 | nM | 8.19 |
| CHEMBL5532322 | — | EC50 | = | 8.309 | nM | 8.08 |
| CHEMBL5568143 | — | EC50 | = | 10.0 | nM | 8.00 |
| CHEMBL5566450 | — | EC50 | = | 18.26 | nM | 7.74 |
| CHEMBL3989767 | CALCITONIN SALMON | EC50 | = | 0.0029 | nM | - |