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Assay Detail

CHEMBL5528176

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antileishmanial activity against Leishmania mexicana intracellular amastigotes infected in J774 macrophages assessed as reduction in parasite viability after 72 hrs by MTT analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Leishmania mexicana
Confidence 1 — Organism
Curated By Autocuration

Target

Leishmania mexicana (CHEMBL612880)
Type ORGANISM
Organism Leishmania mexicana

Publication

Synthetic product-based approach toward potential antileishmanial drug development.
Pal R, Teli G, Akhtar MJ, Matada GSP.
Eur J Med Chem (2024) 263 : 115927 -115927
PubMed 37976706 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.52 7.52

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL7668 1 7.52

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL7668 IC50 = 30.0 nM 7.52