Assay Detail
Functional
CHEMBL5533902
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Antiproliferative activity against mouse MEF cells assessed as cell growth inhibition measured after 48 hrs by MTT assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Cell Type | MEF |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
Dual inhibitors of HDAC and other epigenetic regulators: A novel strategy for cancer treatment.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 5.24 | 5.24 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3989941 | TINOSTAMUSTINE | 2.0 | 1 | 5.24 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3989941 | TINOSTAMUSTINE | IC50 | = | 5700.0 | nM | 5.24 |