Assay Detail
Binding
CHEMBL5537013
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Inhibition of MMP-9 (unknown origin)
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Unveiling sultam in drug discovery: spotlight on the underexplored scaffold.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 8.37 | 9.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL103418 | — | — | 1 | 9.05 |
| CHEMBL103563 | — | — | 1 | 8.07 |
| CHEMBL322433 | — | — | 1 | 8.00 |
| CHEMBL101789 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL103418 | — | Ki | = | 0.9 | nM | 9.05 |
| CHEMBL103563 | — | Ki | = | 8.5 | nM | 8.07 |
| CHEMBL322433 | — | Ki | = | 10.0 | nM | 8.00 |
| CHEMBL101789 | — | Ki | < | 2.1 | nM | - |