Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL5540495

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of KDM5B (unknown origin)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 9 — Direct single protein target
Curated By Autocuration

Target

Lysine-specific demethylase 5B (CHEMBL3774295)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Combination Therapy and Dual-Target Inhibitors Based on LSD1: New Emerging Tools in Cancer Therapy.
Shen L, Wang B, Wang SP, Ji SK, Fu MJ, Wang SW, Hou WQ, Dai XJ, Liu HM.
J Med Chem (2024) 67 : 922 -951
PubMed 38214982 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 8.00 8.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL4454253 1 8.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL4454253 IC50 = 10.0 nM 8.00