Assay Detail
Binding
CHEMBL5541918
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human full length recombinant HIPK4 using RRRFRPASPLRGP as substrate incubated for 120 mins by [33P]-gammaATP based Radiometric scintillation counting analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Homeodomain-interacting protein kinase 4 (CHEMBL1075167) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Discovery and Characterization of Selective, First-in-Class Inhibitors of Citron Kinase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 5.64 | 5.64 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5572737 | — | — | 1 | 5.64 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5572737 | — | IC50 | = | 2275.0 | nM | 5.64 |