Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL5543250

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiinflammatory activity in mouse BV-2 cells assessed as reduction in LPS-induced NO production by Griess reagent based analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Cell Type BV-2
Confidence 1 — Organism
Curated By Autocuration

Target

BV-2 (CHEMBL614781)
Type CELL-LINE
Organism Mus musculus

Publication

Discovery of anti-inflammatory natural flavonoids: Diverse scaffolds and promising leads for drug discovery.
Li J, Zhao R, Miao P, Xu F, Chen J, Jiang X, Hui Z, Wang L, Bai R.
Eur J Med Chem (2023) 260 : 115791 -115791
PubMed 37683361 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 4.57 4.57

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL487601 JACEOSIDINE 1 4.57

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL487601 JACEOSIDINE IC50 = 27000.0 nM 4.57