Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL5543463

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of Hsp70 (unknown origin) by ATPase activity
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Homo sapiens
Confidence 0 — Uncurated / Unknown
Curated By Autocuration

Target

Unchecked (CHEMBL612545)
Type UNCHECKED

Publication

Small molecules targeting molecular chaperones for tau regulation: Achievements and challenges.
He C, Gu J, Wang D, Wang K, Wang Y, You Q, Wang L.
Eur J Med Chem (2023) 261 : 115859 -115859
PubMed 37839344 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 5.90 6.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL470334 1 6.30
CHEMBL5579662 1 5.50

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL470334 IC50 = 500.0 nM 6.30
CHEMBL5579662 IC50 = 3200.0 nM 5.50