Assay Detail
Binding
CHEMBL5545819
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of C57BL/6J mouse Alpha-glucosidase incubated for 10 mins by Lineweaver-Burk plot analysis
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Mus musculus |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Amphiphilic α-Peptoid-deoxynojirimycin Conjugate-based Multivalent Glycosidase Inhibitor for Hypoglycemic Effect and Fluorescence Imaging.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 5.91 | 7.41 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL307429 | DUVOGLUSTAT | 2.0 | 1 | 7.41 |
| CHEMBL1561 | MIGLITOL | 4.0 | 1 | 5.84 |
| CHEMBL5573135 | — | — | 1 | 5.57 |
| CHEMBL5570547 | — | — | 1 | 4.81 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL307429 | DUVOGLUSTAT | Ki | = | 39.0 | nM | 7.41 |
| CHEMBL1561 | MIGLITOL | Ki | = | 1460.0 | nM | 5.84 |
| CHEMBL5573135 | — | Ki | = | 2700.0 | nM | 5.57 |
| CHEMBL5570547 | — | Ki | = | 15400.0 | nM | 4.81 |