Assay Detail
Binding
CHEMBL5548888
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of human recombinant PREP expressed in Escherichia coli BL21 (DE3) cells
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Druglike, <sup>18</sup>F-labeled PET Tracers Targeting Fibroblast Activation Protein.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 5.75 | 5.75 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3233842 | — | — | 1 | 5.75 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3233842 | — | IC50 | = | 1800.0 | nM | 5.75 |