Assay Detail
Binding
CHEMBL5577932
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Binding affinity to N-terminal peptide SR12 of C5aR2 (6 to 32 residues)(unknown origin) assessed as dissociation constant by fluorescence based analysis
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
C5a anaphylatoxin chemotactic receptor 2 (CHEMBL4523478) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Structure of Designer Antibody-like Peptides Binding to the Human C5a with Potential to Modulate the C5a Receptor Signaling.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 2 | 6.69 | 6.69 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5594087 | — | — | 1 | 6.69 |
| CHEMBL5594178 | — | — | 1 | 6.69 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5594087 | — | Kd | = | 203.0 | nM | 6.69 |
| CHEMBL5594178 | — | Kd | = | 203.0 | nM | 6.69 |