Assay Detail
Binding
CHEMBL5579408
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of STT3A/STT3B mediated N-linked glycosylation in human H1-HeLa cells stably transduced with ERluc by measuring effective concentration of inhibition incubated for 18 hrs by One-Glo luciferase reporter assay
25
Total Activities
25
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | H1-HeLa |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Discovery of Potent STT3A/B Inhibitors and Assessment of Their Multipathogen Antiviral Potential and Safety.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 25 | 6.96 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5583975 | — | — | 1 | 9.00 |
| CHEMBL5595779 | — | — | 1 | 8.70 |
| CHEMBL5583748 | — | — | 1 | 8.30 |
| CHEMBL5592276 | — | — | 1 | 8.30 |
| CHEMBL5584184 | — | — | 1 | 7.82 |
| CHEMBL5583722 | — | — | 1 | 7.68 |
| CHEMBL5591147 | — | — | 1 | 7.64 |
| CHEMBL5593281 | — | — | 1 | 7.51 |
| CHEMBL5595895 | — | — | 1 | 7.50 |
| CHEMBL5589992 | — | — | 1 | 7.44 |
| CHEMBL5592540 | — | — | 1 | 7.21 |
| CHEMBL5593163 | — | — | 1 | 6.97 |
| CHEMBL5595968 | — | — | 1 | 6.76 |
| CHEMBL5595888 | — | — | 1 | 6.55 |
| CHEMBL5591248 | — | — | 1 | 6.48 |
| CHEMBL5594134 | — | — | 1 | 6.41 |
| CHEMBL5593573 | — | — | 1 | 6.39 |
| CHEMBL5595336 | — | — | 1 | 6.29 |
| CHEMBL1720448 | — | — | 1 | 6.23 |
| CHEMBL5590333 | — | — | 1 | 6.21 |
| CHEMBL5579784 | — | — | 1 | 6.11 |
| CHEMBL5590068 | — | — | 1 | 6.08 |
| CHEMBL5592058 | — | — | 1 | 5.86 |
| CHEMBL5583718 | — | — | 1 | 5.36 |
| CHEMBL1897966 | — | — | 1 | 5.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5583975 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL5595779 | — | EC50 | = | 2.0 | nM | 8.70 |
| CHEMBL5583748 | — | EC50 | = | 5.0 | nM | 8.30 |
| CHEMBL5592276 | — | EC50 | = | 5.0 | nM | 8.30 |
| CHEMBL5584184 | — | EC50 | = | 15.0 | nM | 7.82 |
| CHEMBL5583722 | — | EC50 | = | 21.0 | nM | 7.68 |
| CHEMBL5591147 | — | EC50 | = | 23.0 | nM | 7.64 |
| CHEMBL5593281 | — | EC50 | = | 31.0 | nM | 7.51 |
| CHEMBL5595895 | — | EC50 | = | 32.0 | nM | 7.50 |
| CHEMBL5589992 | — | EC50 | = | 36.0 | nM | 7.44 |
| CHEMBL5592540 | — | EC50 | = | 62.0 | nM | 7.21 |
| CHEMBL5593163 | — | EC50 | = | 107.0 | nM | 6.97 |
| CHEMBL5595968 | — | EC50 | = | 172.0 | nM | 6.76 |
| CHEMBL5595888 | — | EC50 | = | 279.0 | nM | 6.55 |
| CHEMBL5591248 | — | EC50 | = | 332.0 | nM | 6.48 |
| CHEMBL5594134 | — | EC50 | = | 394.0 | nM | 6.41 |
| CHEMBL5593573 | — | EC50 | = | 409.0 | nM | 6.39 |
| CHEMBL5595336 | — | EC50 | = | 513.0 | nM | 6.29 |
| CHEMBL1720448 | — | EC50 | = | 589.0 | nM | 6.23 |
| CHEMBL5590333 | — | EC50 | = | 615.0 | nM | 6.21 |
| CHEMBL5579784 | — | EC50 | = | 779.0 | nM | 6.11 |
| CHEMBL5590068 | — | EC50 | = | 827.0 | nM | 6.08 |
| CHEMBL5592058 | — | EC50 | = | 1390.0 | nM | 5.86 |
| CHEMBL5583718 | — | EC50 | = | 4420.0 | nM | 5.36 |
| CHEMBL1897966 | — | EC50 | = | 5011.0 | nM | 5.30 |