Assay Detail
Functional
CHEMBL5582734
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of cell proliferation in human A2058 cells incubated for 72 hrs by CellTiter-Glo luminescence assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | A2058 |
| Confidence | 1 — Organism |
| Curated By | Autocuration |
Publication
A Mitochondria-Targeting SIRT3 Inhibitor with Activity against Diffuse Large B Cell Lymphoma.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 5.23 | 5.23 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5595804 | — | — | 1 | 5.23 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5595804 | — | IC50 | = | 5900.0 | nM | 5.23 |