Assay Detail
Binding
CHEMBL5585017
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Inhibition of MPS1 (unknown origin)
16
Total Activities
16
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Hijacking monopolar spindle 1 (MPS1) for various cancer types by small molecular inhibitors: Deep insights from a decade of research and patents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 16 | 8.34 | 9.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL5598395 | — | — | 1 | 9.15 |
| CHEMBL5401292 | — | — | 1 | 9.14 |
| CHEMBL4449557 | — | — | 1 | 9.05 |
| CHEMBL4585148 | — | — | 1 | 9.00 |
| CHEMBL2047959 | — | — | 1 | 8.70 |
| CHEMBL3092039 | — | — | 1 | 8.70 |
| CHEMBL3109945 | — | — | 1 | 8.52 |
| CHEMBL5597789 | — | — | 1 | 8.34 |
| CHEMBL3092037 | — | — | 1 | 8.30 |
| CHEMBL5438574 | — | — | 1 | 8.06 |
| CHEMBL5596286 | — | — | 1 | 8.06 |
| CHEMBL3092036 | — | — | 1 | 8.05 |
| CHEMBL3092035 | — | — | 1 | 7.92 |
| CHEMBL3092030 | — | — | 1 | 7.70 |
| CHEMBL3092029 | — | — | 1 | 7.66 |
| CHEMBL7064 | — | — | 1 | 7.01 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL5598395 | — | IC50 | = | 0.7 | nM | 9.15 |
| CHEMBL5401292 | — | IC50 | = | 0.73 | nM | 9.14 |
| CHEMBL4449557 | — | IC50 | = | 0.9 | nM | 9.05 |
| CHEMBL4585148 | — | IC50 | = | 1.0 | nM | 9.00 |
| CHEMBL2047959 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3092039 | — | IC50 | = | 2.0 | nM | 8.70 |
| CHEMBL3109945 | — | IC50 | = | 3.0 | nM | 8.52 |
| CHEMBL5597789 | — | IC50 | = | 4.6 | nM | 8.34 |
| CHEMBL3092037 | — | IC50 | = | 5.0 | nM | 8.30 |
| CHEMBL5438574 | — | IC50 | = | 8.7 | nM | 8.06 |
| CHEMBL5596286 | — | IC50 | = | 8.7 | nM | 8.06 |
| CHEMBL3092036 | — | IC50 | = | 9.0 | nM | 8.05 |
| CHEMBL3092035 | — | IC50 | = | 12.0 | nM | 7.92 |
| CHEMBL3092030 | — | IC50 | = | 20.0 | nM | 7.70 |
| CHEMBL3092029 | — | IC50 | = | 22.0 | nM | 7.66 |
| CHEMBL7064 | — | IC50 | = | 98.0 | nM | 7.01 |