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Assay Detail

CHEMBL5611084

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Antiviral activity against EBOV Kikwit infected in HeLa cells
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Ebolavirus
Cell Type HeLa
Confidence 1 — Organism
Curated By Autocuration

Target

Ebolavirus (CHEMBL4434621)
Type ORGANISM
Organism Ebolavirus

Publication

Discovery of Thiophene Derivatives as Potent, Orally Bioavailable, and Blood-Brain Barrier-Permeable Ebola Virus Entry Inhibitors.
Morales-Tenorio M, Lasala F, Garcia-Rubia A, Aledavood E, Heung M, Olal C, Escudero-Pérez B, Alonso C, Martínez A, Muñoz-Fontela C, Delgado R, Gil C.
J Med Chem (2024) 67 : 16381 -16402
PubMed 39248591 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 1 4.93 4.93

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL1236524 GALIDESIVIR 2.0 1 4.93

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL1236524 GALIDESIVIR EC50 = 11800.0 nM 4.93