Assay Detail
Binding
CHEMBL5621856
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of recombinant human PDGFRbeta using Poly (Glu,Tyr) 4:1 as substrate incubated for 1 hr by ELISA
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Target
Platelet-derived growth factor receptor beta (CHEMBL1913) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Research progress of VEGFR small molecule inhibitors in ocular neovascular diseases.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 6.94 | 6.94 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4303201 | CATEQUENTINIB | 3.0 | 1 | 6.94 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4303201 | CATEQUENTINIB | IC50 | = | 115.0 | nM | 6.94 |