Assay Detail
Binding
CHEMBL5626276
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Antagonist activity at AR (unknown origin) expressed in chemically activated Luciferase expression system
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Recent advance of small-molecule drugs for clinical treatment of osteoporosis: A review.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 1 | 5.40 | 5.40 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL139835 | CYPROTERONE ACETATE | 3.0 | 1 | 5.40 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL139835 | CYPROTERONE ACETATE | EC50 | = | 4000.0 | nM | 5.40 |