Assay Detail
Binding
CHEMBL5626278
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Displacement of [3H]17 beta estradiol from human ERbeta by radioligand binding assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Recent advance of small-molecule drugs for clinical treatment of osteoporosis: A review.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 7.00 | 7.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL46740 | BAZEDOXIFENE | 4.0 | 1 | 7.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL46740 | BAZEDOXIFENE | IC50 | = | 99.0 | nM | 7.00 |