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Assay Detail

CHEMBL5638463

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Inhibition of Saccharomyces cerevisiae alpha-glucosidase using p-nitrophenyl-alpha-D-glucopyranoside as substrate preincubated for 5 mins followed by substrate addition and measured after 30 mins by spectrophotometric analysis
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Saccharomyces cerevisiae
Confidence 4 — Cell-line / Tissue
Curated By Autocuration

Target

Alpha-glucosidase (CHEMBL5291954)
Type PROTEIN FAMILY
Organism Saccharomyces cerevisiae S288c

Publication

Structural modification of tanshinone IIA and their α-glucosidase inhibitory activity.
Kongphet M, Hang HTX, Ngo TT, Le TK, Chavasiri W.
Bioorg Med Chem Lett (2024) 105 : 129736 -129736
PubMed 38599295 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 7.40 7.40

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL450152 1 7.40

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL450152 IC50 = 40.0 nM 7.40