Assay Detail
Binding
CHEMBL5711488
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of phosphorylated ABL1 Q252H mutant (unknown origin) in presence of ATP by enzymatic assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Pharmacological targeting of kinases MST1 and MST2 augments tissue repair and regeneration.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 7.94 | 7.94 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL4554938 | — | — | 1 | 7.94 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL4554938 | — | IC50 | = | 11.6 | nM | 7.94 |