Assay Detail
Binding
CHEMBL5712155
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of M2 receptor (unknown origin) by radioligand binding assay
1
Total Activities
1
Compounds Tested
1
Activity Types
2
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Discovery of a chemical probe for the L3MBTL3 methyllysine reader domain.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 7.14 | 7.14 |
Assay Parameters
| Parameter | Type | Value | Units | Text |
|---|---|---|---|---|
| EFO_ID | EFO_ID | - | — | EFO:0000616 |
| EFO_TERM | EFO_TERM | - | — | neoplasm |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2426364 | — | — | 1 | 7.14 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2426364 | — | Ki | = | 72.0 | nM | 7.14 |