Assay Detail
Binding
CHEMBL615301
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Binding affinity on 3 beta-hydroxysteroid dehydrogenase
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
3 beta-hydroxysteroid dehydrogenase/Delta 5-->4-isomerase type 1 (CHEMBL1958) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
Pharmacological options in the treatment of benign prostatic hyperplasia.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.45 | 8.08 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL24033 | — | — | 1 | 8.08 |
| CHEMBL24729 | — | — | 1 | 6.82 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL24033 | — | IC50 | = | 8.3 | nM | 8.08 |
| CHEMBL24729 | — | IC50 | = | 150.0 | nM | 6.82 |