Assay Detail
Binding
CHEMBL616378
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Binding affinity for 5-hydroxytryptamine 1A receptor was determined
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Conformationally restricted indolopiperidine derivatives as potent CCR2B receptor antagonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 6.05 | 7.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL432713 | — | — | 1 | 7.00 |
| CHEMBL71707 | — | — | 1 | 5.10 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL432713 | — | Ki | = | 100.0 | nM | 7.00 |
| CHEMBL71707 | — | Ki | = | 7943.28 | nM | 5.10 |