Assay Detail
Binding
CHEMBL616382
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Compound was evaluated for the affinity at 5-hydroxytryptamine 1A receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Selective, orally active 5-HT1D receptor agonists as potential antimigraine agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.81 | 7.26 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL292779 | — | — | 1 | 7.26 |
| CHEMBL128 | SUMATRIPTAN | 4.0 | 1 | 6.35 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL292779 | — | IC50 | = | 55.0 | nM | 7.26 |
| CHEMBL128 | SUMATRIPTAN | IC50 | = | 450.0 | nM | 6.35 |