Assay Detail
Binding
CHEMBL616684
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Ability to displace [3H]-8-OH-DPAT from rat hippocampal homogenate 5-hydroxytryptamine 1A receptor
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Tissue | Hippocampus |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Dihydrobenzofuran analogues of hallucinogens. 4. Mescaline derivatives.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 5.18 | 5.21 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL102347 | — | — | 1 | 5.21 |
| CHEMBL319415 | — | — | 1 | 5.16 |
| CHEMBL26687 | MESCALINE | 1.0 | 1 | 5.16 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL102347 | — | Ki | = | 6200.0 | nM | 5.21 |
| CHEMBL319415 | — | Ki | = | 6900.0 | nM | 5.16 |
| CHEMBL26687 | MESCALINE | Ki | = | 6900.0 | nM | 5.16 |