Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL617303

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Selectivity towards 5-hydroxytryptamine 1D receptor beta to that of 5-hydroxytryptamine 1D receptor alpha
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

5-hydroxytryptamine receptor 1D (CHEMBL1983)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Binding of O-alkyl derivatives of serotonin at human 5-HT1D beta receptors.
Glennon RA, Hong SS, Bondarev M, Law H, Dukat M, Rakhi S, Power P, Fan E, Kinneau D, Kamboj R, Teitler M, Herrick-Davis K, Smith C.
J Med Chem (1996) 39 : 314 -322
PubMed 8568822 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 8.27 8.27

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL8165 5-METHOXYTRYPTAMINE 1 8.27

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL8165 5-METHOXYTRYPTAMINE Ki = 5.4 nM 8.27