Assay Detail
Functional
CHEMBL640252
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Compound was evaluated for the Adenosine A1 receptor agonist potency.
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Cricetulus griseus |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
The design and synthesis of novel adenosine agonists
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 3 | 8.94 | 9.72 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL68738 | N6-CYCLOPENTYLADENOSINE | — | 1 | 9.72 |
| CHEMBL2364570 | — | — | 1 | 9.09 |
| CHEMBL2364571 | — | — | 1 | 8.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL68738 | N6-CYCLOPENTYLADENOSINE | EC50 | = | 0.19 | nM | 9.72 |
| CHEMBL2364570 | — | EC50 | = | 0.81 | nM | 9.09 |
| CHEMBL2364571 | — | EC50 | = | 10.0 | nM | 8.00 |