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Assay Detail

CHEMBL643553

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Binding
In vitro inhibition of Adenosine kinase (AK)
21
Total Activities
21
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Expert

Target

Adenosine kinase (CHEMBL2384)
Type SINGLE PROTEIN
Organism Rattus norvegicus

Publication

Discovery of 4-amino-5-(3-bromophenyl)-7-(6-morpholino-pyridin-3-yl)pyrido[2,3-d]pyrimidine, an orally active, non-nucleoside adenosine kinase inhibitor..
Lee CH, Jiang M, Cowart M, Gfesser G, Perner R, Kim KH, Gu YG, Williams M, Jarvis MF, Kowaluk EA, Stewart AO, Bhagwat SS.
J Med Chem (2001) 44 : 2133 -2138
PubMed 11405650 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 21 7.14 8.80

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL66280 5-IODO,5'-DEOXYTUBERCIDIN 1 8.80
CHEMBL66089 1 8.77
CHEMBL68748 1 8.74
CHEMBL66277 1 8.55
CHEMBL68749 1 8.30
CHEMBL68492 1 8.15
CHEMBL302921 1 8.08
CHEMBL302376 1 7.82
CHEMBL305746 1 7.60
CHEMBL66568 1 7.20
CHEMBL416498 1 7.18
CHEMBL66977 1 7.13
CHEMBL302938 1 7.04
CHEMBL65852 1 6.40
CHEMBL66338 1 6.36
CHEMBL303499 1 6.11
CHEMBL67043 1 5.76
CHEMBL304179 1 5.70
CHEMBL67267 1 5.70
CHEMBL308008 1 5.32
CHEMBL419063 1 5.26

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL66280 5-IODO,5'-DEOXYTUBERCIDIN IC50 = 1.6 nM 8.80
CHEMBL66089 IC50 = 1.7 nM 8.77
CHEMBL68748 IC50 = 1.8 nM 8.74
CHEMBL66277 IC50 = 2.8 nM 8.55
CHEMBL68749 IC50 = 5.0 nM 8.30
CHEMBL68492 IC50 = 7.0 nM 8.15
CHEMBL302921 IC50 = 8.3 nM 8.08
CHEMBL302376 IC50 = 15.0 nM 7.82
CHEMBL305746 IC50 = 25.0 nM 7.60
CHEMBL66568 IC50 = 62.5 nM 7.20
CHEMBL416498 IC50 = 66.7 nM 7.18
CHEMBL66977 IC50 = 73.3 nM 7.13
CHEMBL302938 IC50 = 91.7 nM 7.04
CHEMBL65852 IC50 = 400.0 nM 6.40
CHEMBL66338 IC50 = 440.0 nM 6.36
CHEMBL303499 IC50 = 773.0 nM 6.11
CHEMBL67043 IC50 = 1750.0 nM 5.76
CHEMBL304179 IC50 = 2000.0 nM 5.70
CHEMBL67267 IC50 = 2000.0 nM 5.70
CHEMBL308008 IC50 = 4750.0 nM 5.32
CHEMBL419063 IC50 = 5500.0 nM 5.26