Assay Detail
Binding
CHEMBL645553
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Compound was evaluated for binding affinity against Alpha-1 adrenergic receptor from rat
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 4 — Cell-line / Tissue |
| Curated By | Autocuration |
Publication
NGB 2904 and NGB 2849: two highly selective dopamine D3 receptor antagonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 6.23 | 6.26 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL419505 | — | — | 1 | 6.26 |
| CHEMBL300780 | — | — | 1 | 6.19 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL419505 | — | Ki | = | 547.0 | nM | 6.26 |
| CHEMBL300780 | — | Ki | = | 642.0 | nM | 6.19 |