Assay Detail
Functional
CHEMBL646296
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonistic activity against Alpha-1 adrenergic receptor in the epidermal portion of the rat vas deferens
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Tissue | Vas deferens |
| Confidence | 4 — Cell-line / Tissue |
| Curated By | Autocuration |
Publication
Structure-activity relationships for 2-substituted imidazoles as alpha 2-adrenoceptor antagonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 2 | 5.00 | 5.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1203734 | — | — | 1 | 5.00 |
| CHEMBL1203738 | — | — | 1 | 5.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1203734 | — | Kd | = | 10000.0 | nM | 5.00 |
| CHEMBL1203738 | — | Kd | = | 10000.0 | nM | 5.00 |