Assay Detail
Binding
CHEMBL646480
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Binding affinity for adenosine A2 receptor using [3H]- NECA
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Rattus norvegicus |
| Confidence | 5 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Publication
Adenosine receptors: pharmacology, structure-activity relationships, and therapeutic potential.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 8.62 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL610440 | — | — | 1 | 9.00 |
| CHEMBL1950647 | — | — | 1 | 8.24 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL610440 | — | Ki | = | 1.0 | nM | 9.00 |
| CHEMBL1950647 | — | Ki | = | 5.7 | nM | 8.24 |