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Assay Detail

CHEMBL648099

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
The compound was tested for binding affinity against Alpha-1B adrenergic receptor, from hamster clones.
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Cricetulus griseus
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Alpha-1B adrenergic receptor (CHEMBL232)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Alpha- and beta-adrenoceptors: from the gene to the clinic. 1. Molecular biology and adrenoceptor subclassification.
Hieble JP, Bondinell WE, Ruffolo RR.
J Med Chem (1995) 38 : 3415 -3444
PubMed 7658428 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 7.60 7.60

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL279516 INDORAMIN 2.0 1 7.60

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL279516 INDORAMIN Ki = 25.0 nM 7.60