Assay Detail
Binding
CHEMBL648319
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In vitro beta adrenergic receptor blocking in guinea pig trachea
2
Total Activities
2
Compounds Tested
2
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Cavia porcellus |
| Tissue | Trachea |
| Confidence | 4 — Cell-line / Tissue |
| Curated By | Autocuration |
Publication
[(Arylcarbonyl)oxy]propanolamines. 1. Novel beta-blockers with ultrashort duration of action.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 1 | 8.20 | 8.20 |
| pA2 | 1 | - | - |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL6935 | — | — | 1 | 8.20 |
| CHEMBL7509 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL6935 | — | Kd | = | 6.31 | nM | 8.20 |
| CHEMBL7509 | — | pA2 | - | — | - |