Assay Detail
Binding
CHEMBL648324
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity against GST-hARLBD was measured in SC-3 cell by using [3H]testosterone as radioligand
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Cell Type | SC-3 |
| Confidence | 9 — Direct single protein target |
| Curated By | Expert |
Publication
Anti-androgens with full antagonistic activity toward human prostate tumor LNCaP cells with mutated androgen receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 5.89 | 5.89 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL806 | FLUTAMIDE | 4.0 | 1 | 5.89 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL806 | FLUTAMIDE | Ki | = | 1300.0 | nM | 5.89 |