Assay Detail
Binding
CHEMBL649645
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of [3H]- rauwolscine binding to alpha-2 adrenergic receptor in rat cerebral cortex
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Tissue | Cerebral cortex |
| Confidence | 4 — Cell-line / Tissue |
| Curated By | Autocuration |
Publication
New potential uroselective NO-donor alpha1-antagonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 7.48 | 7.48 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL278865 | UPIDOSIN | 2.0 | 1 | 7.48 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL278865 | UPIDOSIN | Ki | = | 33.3 | nM | 7.48 |