Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL649975

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Inhibition of chemotactic protein to CCR5
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

C-C chemokine receptor type 5 (CHEMBL274)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Inhibition of protein-protein association by small molecules: approaches and progress.
Toogood PL.
J Med Chem (2002) 45 : 1543 -1558
PubMed 11931608 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 8.92 8.92

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL41275 1 8.92

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL41275 IC50 = 1.2 nM 8.92