Assay Detail
Binding
CHEMBL649989
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibitory activity against TEM-1 Beta-lactamase mutant G238A at 42 degree Centigrade
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Escherichia coli |
| Confidence | 9 — Direct single protein target |
| Curated By | Intermediate |
Publication
A specific mechanism of nonspecific inhibition.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 5.16 | 5.16 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1160008 | IODOPHTHALEIN | 2.0 | 1 | 5.16 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1160008 | IODOPHTHALEIN | IC50 | = | 7000.0 | nM | 5.16 |