Assay Detail
Binding
CHEMBL650505
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Compound was tested for its ability to inhibit C-C chemokine receptor type 3 receptor
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Design and synthesis of novel CCR3 antagonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 4 | 8.31 | 8.62 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL431670 | — | — | 1 | 8.62 |
| CHEMBL121637 | — | — | 1 | 8.36 |
| CHEMBL121905 | — | — | 1 | 8.33 |
| CHEMBL436363 | — | — | 1 | 7.92 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL431670 | — | IC50 | = | 2.4 | nM | 8.62 |
| CHEMBL121637 | — | IC50 | = | 4.4 | nM | 8.36 |
| CHEMBL121905 | — | IC50 | = | 4.7 | nM | 8.33 |
| CHEMBL436363 | — | IC50 | = | 12.0 | nM | 7.92 |