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Assay Detail

CHEMBL650903

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity at C-C chemokine receptor type 5
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

C-C chemokine receptor type 5 (CHEMBL274)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Piperazine-based CCR5 antagonists as HIV-1 inhibitors. II. Discovery of 1-[(2,4-dimethyl-3-pyridinyl)carbonyl]-4- methyl-4-[3(S)-methyl-4-[1(S)-[4-(trifluoromethyl)phenyl]ethyl]-1-piperazinyl]- piperidine N1-oxide (Sch-350634), an orally bioavailable, potent CCR5 antagonist.
Tagat JR, Steensma RW, McCombie SW, Nazareno DV, Lin SI, Neustadt BR, Cox K, Xu S, Wojcik L, Murray MG, Vantuno N, Baroudy BM, Strizki JM.
J Med Chem (2001) 44 : 3343 -3346
PubMed 11585438 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 2 8.40 8.64

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL113436 1 8.64
CHEMBL322251 1 8.15

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL113436 Ki = 2.3 nM 8.64
CHEMBL322251 Ki = 7.0 nM 8.15