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Assay Detail

CHEMBL651754

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Effect of compound against Moloney murine sarcoma virus (MSV)-induced transformation of C3H/3T3 embryo murine fibroblasts
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Cell Type C3H/3T3
Confidence 1 — Organism
Curated By Intermediate

Target

C3H/3T3 (CHEMBL614372)
Type CELL-LINE
Organism Mus musculus

Publication

cycloSal-Pronucleotides of 2',3'-dideoxyadenosine and 2', 3'-dideoxy-2',3'-didehydroadenosine: synthesis and antiviral evaluation of a highly efficient nucleotide delivery system.
Meier C, Knispel T, De Clercq E, Balzarini J.
J Med Chem (1999) 42 : 1604 -1614
PubMed 10229629 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 3 5.63 5.93

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL40302 1 5.93
CHEMBL416624 1 5.54
CHEMBL289937 1 5.41

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL40302 EC50 = 1180.0 nM 5.93
CHEMBL416624 EC50 = 2860.0 nM 5.54
CHEMBL289937 EC50 = 3900.0 nM 5.41