Assay Detail
Binding
CHEMBL651998
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The compound was tested for binding affinity against Alpha-1B adrenergic receptor, from human clones.
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Alpha- and beta-adrenoceptors: from the gene to the clinic. 1. Molecular biology and adrenoceptor subclassification.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 7.29 | 7.54 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL279516 | INDORAMIN | 2.0 | 1 | 7.54 |
| CHEMBL420060 | — | — | 1 | 7.04 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL279516 | INDORAMIN | Ki | = | 29.0 | nM | 7.54 |
| CHEMBL420060 | — | Ki | = | 92.0 | nM | 7.04 |