Assay Detail
Functional
CHEMBL652014
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity towards human Beta-3 adrenergic receptor
26
Total Activities
26
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Discovery of L-755,507: a subnanomolar human beta 3 adrenergic receptor agonist.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 26 | 8.61 | 9.37 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL12998 | L-755507 | — | 1 | 9.37 |
| CHEMBL13389 | — | — | 1 | 9.15 |
| CHEMBL13132 | — | — | 1 | 9.00 |
| CHEMBL13467 | — | — | 1 | 9.00 |
| CHEMBL275511 | — | — | 1 | 8.96 |
| CHEMBL12911 | — | — | 1 | 8.96 |
| CHEMBL13068 | — | — | 1 | 8.92 |
| CHEMBL275291 | — | — | 1 | 8.92 |
| CHEMBL268289 | — | — | 1 | 8.85 |
| CHEMBL12943 | — | — | 1 | 8.85 |
| CHEMBL13398 | — | — | 1 | 8.85 |
| CHEMBL13432 | — | — | 1 | 8.72 |
| CHEMBL274144 | — | — | 1 | 8.68 |
| CHEMBL417250 | — | — | 1 | 8.64 |
| CHEMBL13521 | — | — | 1 | 8.62 |
| CHEMBL13106 | — | — | 1 | 8.59 |
| CHEMBL144870 | — | — | 1 | 8.55 |
| CHEMBL12864 | — | — | 1 | 8.34 |
| CHEMBL273428 | — | — | 1 | 8.30 |
| CHEMBL13459 | — | — | 1 | 8.28 |
| CHEMBL417613 | — | — | 1 | 8.20 |
| CHEMBL274143 | — | — | 1 | 8.18 |
| CHEMBL13453 | — | — | 1 | 8.17 |
| CHEMBL275114 | — | — | 1 | 8.00 |
| CHEMBL12939 | — | — | 1 | 7.96 |
| CHEMBL274312 | — | — | 1 | 7.77 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL12998 | L-755507 | EC50 | = | 0.43 | nM | 9.37 |
| CHEMBL13389 | — | EC50 | = | 0.7 | nM | 9.15 |
| CHEMBL13132 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL13467 | — | EC50 | = | 1.0 | nM | 9.00 |
| CHEMBL275511 | — | EC50 | = | 1.1 | nM | 8.96 |
| CHEMBL12911 | — | EC50 | = | 1.1 | nM | 8.96 |
| CHEMBL13068 | — | EC50 | = | 1.2 | nM | 8.92 |
| CHEMBL275291 | — | EC50 | = | 1.2 | nM | 8.92 |
| CHEMBL268289 | — | EC50 | = | 1.4 | nM | 8.85 |
| CHEMBL12943 | — | EC50 | = | 1.4 | nM | 8.85 |
| CHEMBL13398 | — | EC50 | = | 1.4 | nM | 8.85 |
| CHEMBL13432 | — | EC50 | = | 1.9 | nM | 8.72 |
| CHEMBL274144 | — | EC50 | = | 2.1 | nM | 8.68 |
| CHEMBL417250 | — | EC50 | = | 2.3 | nM | 8.64 |
| CHEMBL13521 | — | EC50 | = | 2.4 | nM | 8.62 |
| CHEMBL13106 | — | EC50 | = | 2.6 | nM | 8.59 |
| CHEMBL144870 | — | EC50 | = | 2.8 | nM | 8.55 |
| CHEMBL12864 | — | EC50 | = | 4.6 | nM | 8.34 |
| CHEMBL273428 | — | EC50 | = | 5.0 | nM | 8.30 |
| CHEMBL13459 | — | EC50 | = | 5.2 | nM | 8.28 |
| CHEMBL417613 | — | EC50 | = | 6.3 | nM | 8.20 |
| CHEMBL274143 | — | EC50 | = | 6.6 | nM | 8.18 |
| CHEMBL13453 | — | EC50 | = | 6.8 | nM | 8.17 |
| CHEMBL275114 | — | EC50 | = | 10.0 | nM | 8.00 |
| CHEMBL12939 | — | EC50 | = | 11.0 | nM | 7.96 |
| CHEMBL274312 | — | EC50 | = | 17.0 | nM | 7.77 |