Assay Detail
Binding
CHEMBL652026
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity towards antiestrogen binding site AEBS
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 6 — Multiple protein complex / RNA |
| Curated By | Expert |
Target
Anti-estrogen binding site (AEBS) (CHEMBL612409) ↗| Type | PROTEIN COMPLEX |
| Organism | Homo sapiens |
Publication
Antiestrogens and selective estrogen receptor modulators as multifunctional medicines. 1. Receptor interactions.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 1 | 9.00 | 9.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL83 | TAMOXIFEN | 4.0 | 1 | 9.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL83 | TAMOXIFEN | Kd | = | 1.0 | nM | 9.00 |