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Assay Detail

CHEMBL653137

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Equilibrium dissociation constant (KD) against beta adrenergic receptor of rat lung tissue
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 4 — Cell-line / Tissue
Curated By Autocuration

Target

Adrenergic receptor beta (CHEMBL2095166)
Type PROTEIN FAMILY
Organism Rattus norvegicus

Publication

Alkylating beta-blockers: activity of isomeric bromoacetyl alprenolol menthanes.
Liptak A, Kusiak JW, Pitha J.
J Med Chem (1985) 28 : 1699 -1703
PubMed 2866247 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 1 7.53 7.53

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL46136 BROMOACETYL ALPRENOLOL MENTHANE 1 7.53

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL46136 BROMOACETYL ALPRENOLOL MENTHANE Kd = 29.3 nM 7.53