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Assay Detail

CHEMBL653537

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Functional
Effective concentration required to inhibit the replication of HIV-1 in CEMSS human T4 lymphoblastoid cell lines
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type CEM-SS
Confidence 1 — Organism
Curated By Intermediate

Target

CEM-SS (CHEMBL614548)
Type CELL-LINE
Organism Homo sapiens

Publication

Increase of the adenallene anti-HIV activity in cell culture using its bis(tBuSATE) phosphotriester derivative.
Egron D, Périgaud C, Gosselin G, Aubertin AM, Gatanaga H, Mitsuya H, Zemlicka J, Imbach JL.
Bioorg Med Chem Lett (2002) 12 : 265 -266
PubMed 11755368 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
EC50 2 5.09 5.92

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL264014 1 5.92
CHEMBL313478 1 4.25

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL264014 EC50 = 1200.0 nM 5.92
CHEMBL313478 EC50 = 56000.0 nM 4.25